PT-141 (Bremelanotide)

Home

Peptide Clinic

Peptide Clinic

PT-141 (Bremelanotide)

Product Description

Strength and Packaging:
PT-141 (Bremelanotide) is typically provided in a 10 ml vial with a concentration of 1 mg per ml, totaling 10 mg per vial. This concentration is optimal for precise dosing, catering to both occasional and regular use for its intended purposes.

Molecular Structure:

Molecular Formula: C50H68N14O10
Molecular Weight: 1025.2 g/mol
Sequence: Ac-Nle-cyclo(Asp-His-D-Phe-Arg-Trp-Lys)-OH

Function and Purpose:
PT-141, also known as Bremelanotide, is a synthetic peptide developed from Melanotan II, primarily used to treat sexual dysfunction in both men (erectile dysfunction) and women (hypoactive sexual desire disorder). Unlike other sexual dysfunction treatments, PT-141 does not act on the vascular system but directly affects the nervous system by activating melanocortin receptors.

Cellular Mechanism of Action:

Activation of Melanocortin Receptors: PT-141 works by stimulating melanocortin receptors, particularly MC3-R and MC4-R, located in the central nervous system. These receptors are involved in regulating sexual arousal and desire.
Neurogenic Action: By bypassing the vascular system and acting directly on the brain's arousal centers, PT-141 triggers sexual arousal in both men and women.
Influence on Sexual Pathways: It enhances the sexual response by promoting dopamine release, a neurotransmitter critical for sexual arousal and pleasure.

Effects on the Body:
PT-141 primarily enhances sexual arousal and desire without affecting systemic blood pressure, making it a unique treatment option for sexual dysfunctions. It also influences the psychological and physiological pathways that regulate libido and sexual performance.

Order Now

Improves Sexual Arousal: Directly stimulates sexual desire and arousal by acting on the central nervous system.
Treats Erectile Dysfunction: Effective in men who do not respond to other erectile dysfunction medications like PDE5 inhibitors (e.g., Viagra, Cialis).
Addresses Female Sexual Dysfunction: Proven to enhance sexual desire and arousal in women with hypoactive sexual desire disorder (HSDD).
Non-Systemic Action: Unlike other sexual enhancement drugs, it does not affect cardiovascular function, making it safer for individuals with certain health conditions.
Quick Onset: Provides rapid effects, usually within 30-60 minutes after administration.

Targeted Conditions and Health Goals:

Treatment of erectile dysfunction (ED) in men
Enhancing sexual desire and arousal in women with HSDD
Alternative for individuals who cannot use traditional PDE5 inhibitors

Study 1: Journal of Sexual Medicine reported that PT-141 effectively increases sexual arousal in premenopausal women with HSDD, with significant improvements in sexual desire scores.
Study 2: International Journal of Impotence Research demonstrated PT-141's efficacy in treating erectile dysfunction in men who are unresponsive to traditional ED medications, showing substantial improvements in erectile function.
Study 3: Research published in Pharmacology Biochemistry and Behavior highlighted PT-141's unique mechanism of action on the melanocortin system, differentiating it from other ED treatments that primarily target the vascular system.

Additional Findings:

Safety Profile: Clinical trials confirm that PT-141 is well-tolerated, with minimal side effects, particularly for individuals with cardiovascular concerns.
Psychological Benefits: Beyond physical arousal, PT-141 also positively affects mood and mental outlook related to sexual activity.

These studies provide robust evidence supporting PT-141’s role as an effective treatment for sexual dysfunctions, enhancing both physiological and psychological aspects of sexual health.

Recommended Dosage: For most users, the recommended dose of PT-141 is 1-2 mg, administered subcutaneously approximately 30-60 minutes before anticipated sexual activity. Dosage may be adjusted based on individual response and tolerance.
Administration Method: PT-141 is administered via subcutaneous injection, typically in the abdominal or thigh area for optimal absorption.
Frequency and Duration: PT-141 can be used on an as-needed basis, depending on the frequency of sexual activity. It is not intended for daily use but rather on an intermittent schedule tailored to individual needs.

Usage Tips:

Start with a lower dose (1 mg) to assess tolerance.
Avoid using PT-141 more than once within a 24-hour period to prevent potential side effects.

Reconstitution: PT-141 comes pre-reconstituted in a 10 ml vial, ready for immediate use. No additional mixing is required. Simply draw the desired dosage using an insulin syringe.
Storage: Store PT-141 in the refrigerator (2-8°C) in its original packaging to maintain stability and potency. Do not freeze. The product is shipped in cold packing to ensure it remains at the optimal temperature during transit.

Handling Precautions:

Keep the vial in a cool, dark place to protect from light exposure.
Ensure sterile conditions when drawing the peptide to prevent contamination.

Potential Side Effects:

Mild nausea, particularly with higher doses.
Possible flushing or a sensation of warmth.
Headaches or dizziness in some users.
Rare instances of increased blood pressure.

Precautions:

Not recommended for pregnant or breastfeeding women.
Individuals with cardiovascular conditions should consult a healthcare provider before use due to potential changes in blood pressure.
Avoid using in conjunction with alcohol or recreational drugs, which may amplify side effects.

Usage Recommendations:

Users should be aware of their personal tolerance levels and adjust dosages accordingly.
PT-141 should not be used by individuals with a known allergy to any of its components.

What is PT-141, and how does it work?
PT-141, or Bremelanotide, is a synthetic peptide that stimulates melanocortin receptors in the brain to enhance sexual arousal and desire.
How should I use PT-141?
Administer PT-141 via subcutaneous injection approximately 30-60 minutes before sexual activity.
Are there any side effects?
Some users may experience mild nausea, flushing, or headaches. These side effects are generally short-lived.
Can I use PT-141 if I have heart conditions?
Consult with a healthcare provider before use if you have cardiovascular conditions, as PT-141 can affect blood pressure.
Is PT-141 suitable for both men and women?
Yes, PT-141 is effective for treating sexual dysfunction in both men and women.
How often can I use PT-141?
PT-141 is intended for use on an as-needed basis and should not be used more than once within a 24-hour period.

Purity and Quality: Our PT-141 is synthesized in a GMP-certified facility, ensuring the highest standards of purity and quality.
Third-Party Testing: Each batch undergoes rigorous third-party testing to verify purity levels (>99%) and ensure it is free from contaminants.
Certifications and Transparency: Certificates of Analysis (COA) are available upon request, offering full transparency on product quality.

Shipping: We offer worldwide shipping with tracking. Orders are processed within 1-2 business days, and express shipping options are available.
Cold Packing: All PT-141 shipments are packed in cold packaging to maintain product integrity during transit.
Returns: We offer a 30-day return policy on unopened vials. If you are not satisfied with your purchase, please contact customer service for a return authorization.

Suggested Pricing and Purchase Options

10 ml Vial (1 mg/ml): $129.99 USD
Bulk Purchase Discount: Buy 3 vials for $359.99 USD (Save $30)
Subscription Offer: Subscribe and save 15% on all orders with a monthly auto-ship program.

Customer Service and Bulk Orders:
For large orders or personalized dosage recommendations, please contact our customer service team. They are available to help customize your order and ensure you receive the best pricing and product guidance.

Order Now

Reviews and Testimonials

"PT-141 has transformed my sex life. I’ve noticed a significant increase in arousal and desire. It’s a great alternative to traditional ED medications."

Mark L.

"As a woman struggling with low libido, PT-141 has been a game-changer. It’s helped me feel more connected and confident in my intimate moments."

Laura K.

"This peptide works quickly and effectively. I’ve tried many treatments, and PT-141 is by far the best for my needs."

Kevin T.

Related Products

Peptide Clinic

Melanotan II

View Details