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PT-141 (Bremelanotide) is typically provided in a 10 ml vial with a concentration of 1 mg per ml, totaling 10 mg per vial. This concentration is optimal for precise dosing, catering to both occasional and regular use for its intended purposes.
Estimated Delivery:7 days
Shipping Charge:
$ 60
Product Description
Strength and Packaging:
PT-141 (Bremelanotide) is typically provided in a 10 ml vial with a concentration of 1 mg per ml, totaling 10 mg per vial. This concentration is optimal for precise dosing, catering to both occasional and regular use for its intended purposes.
Molecular Structure: Molecular Formula: C50H68N14O10 Molecular Weight: 1025.2 g/mol Sequence: Ac-Nle-cyclo(Asp-His-D-Phe-Arg-Trp-Lys)-OH
Function and Purpose:
PT-141, also known as Bremelanotide, is a synthetic peptide developed from Melanotan II, primarily used to treat sexual dysfunction in both men (erectile dysfunction) and women (hypoactive sexual desire disorder). Unlike other sexual dysfunction treatments, PT-141 does not act on the vascular system but directly affects the nervous system by activating melanocortin receptors.
Cellular Mechanism of Action:
Activation of Melanocortin Receptors: PT-141 works by stimulating melanocortin receptors, particularly MC3-R and MC4-R, located in the central nervous system. These receptors are involved in regulating sexual arousal and desire.
Neurogenic Action: By bypassing the vascular system and acting directly on the brain's arousal centers, PT-141 triggers sexual arousal in both men and women.
Influence on Sexual Pathways: It enhances the sexual response by promoting dopamine release, a neurotransmitter critical for sexual arousal and pleasure.
Effects on the Body:
Shipping: We offer worldwide shipping with tracking. Orders are processed within 1-2 business days, and express shipping options are available.
Cold Packing: All PT-141 shipments are packed in cold packaging to maintain product integrity during transit.
Returns: We offer a 30-day return policy on unopened vials. If you are not satisfied with your purchase, please contact customer service for a return authorization.
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Improves Sexual Arousal: Directly stimulates sexual desire and arousal by acting on the central nervous system.
Treats Erectile Dysfunction: Effective in men who do not respond to other erectile dysfunction medications like PDE5 inhibitors (e.g., Viagra, Cialis).
Addresses Female Sexual Dysfunction: Proven to enhance sexual desire and arousal in women with hypoactive sexual desire disorder (HSDD).
Non-Systemic Action: Unlike other sexual enhancement drugs, it does not affect cardiovascular function, making it safer for individuals with certain health conditions.
Quick Onset: Provides rapid effects, usually within 30-60 minutes after administration.
Targeted Conditions and Health Goals:
Treatment of erectile dysfunction (ED) in men
Enhancing sexual desire and arousal in women with HSDD
Alternative for individuals who cannot use traditional PDE5 inhibitors
Study 1: Journal of Sexual Medicine reported that PT-141 effectively increases sexual arousal in premenopausal women with HSDD, with significant improvements in sexual desire scores.
Study 2: International Journal of Impotence Research demonstrated PT-141's efficacy in treating erectile dysfunction in men who are unresponsive to traditional ED medications, showing substantial improvements in erectile function.
Study 3: Research published in Pharmacology Biochemistry and Behavior highlighted PT-141's unique mechanism of action on the melanocortin system, differentiating it from other ED treatments that primarily target the vascular system.
Additional Findings:
Safety Profile: Clinical trials confirm that PT-141 is well-tolerated, with minimal side effects, particularly for individuals with cardiovascular concerns.
Psychological Benefits: Beyond physical arousal, PT-141 also positively affects mood and mental outlook related to sexual activity.
These studies provide robust evidence supporting PT-141’s role as an effective treatment for sexual dysfunctions, enhancing both physiological and psychological aspects of sexual health.
Recommended Dosage: For most users, the recommended dose of PT-141 is 1-2 mg, administered subcutaneously approximately 30-60 minutes before anticipated sexual activity. Dosage may be adjusted based on individual response and tolerance.
Administration Method: PT-141 is administered via subcutaneous injection, typically in the abdominal or thigh area for optimal absorption.
Frequency and Duration: PT-141 can be used on an as-needed basis, depending on the frequency of sexual activity. It is not intended for daily use but rather on an intermittent schedule tailored to individual needs.
Usage Tips:
Start with a lower dose (1 mg) to assess tolerance.
Avoid using PT-141 more than once within a 24-hour period to prevent potential side effects.
Reconstitution: PT-141 comes pre-reconstituted in a 10 ml vial, ready for immediate use. No additional mixing is required. Simply draw the desired dosage using an insulin syringe.
Storage: Store PT-141 in the refrigerator (2-8°C) in its original packaging to maintain stability and potency. Do not freeze. The product is shipped in cold packing to ensure it remains at the optimal temperature during transit.
Handling Precautions:
Keep the vial in a cool, dark place to protect from light exposure.
Ensure sterile conditions when drawing the peptide to prevent contamination.
Potential Side Effects: Mild nausea, particularly with higher doses. Possible flushing or a sensation of warmth. Headaches or dizziness in some users. Rare instances of increased blood pressure.
Precautions: Not recommended for pregnant or breastfeeding women. Individuals with cardiovascular conditions should consult a healthcare provider before use due to potential changes in blood pressure. Avoid using in conjunction with alcohol or recreational drugs, which may amplify side effects.
Usage Recommendations: Users should be aware of their personal tolerance levels and adjust dosages accordingly. PT-141 should not be used by individuals with a known allergy to any of its components.
What is PT-141, and how does it work?
PT-141, or Bremelanotide, is a synthetic peptide that stimulates melanocortin receptors in the brain to enhance sexual arousal and desire.
How should I use PT-141?
Administer PT-141 via subcutaneous injection approximately 30-60 minutes before sexual activity.
Are there any side effects?
Some users may experience mild nausea, flushing, or headaches. These side effects are generally short-lived.
Can I use PT-141 if I have heart conditions?
Consult with a healthcare provider before use if you have cardiovascular conditions, as PT-141 can affect blood pressure.
Is PT-141 suitable for both men and women?
Yes, PT-141 is effective for treating sexual dysfunction in both men and women.
How often can I use PT-141?
PT-141 is intended for use on an as-needed basis and should not be used more than once within a 24-hour period.
Purity and Quality: Our PT-141 is synthesized in a GMP-certified facility, ensuring the highest standards of purity and quality.
Third-Party Testing: Each batch undergoes rigorous third-party testing to verify purity levels (>99%) and ensure it is free from contaminants.
Certifications and Transparency: Certificates of Analysis (COA) are available upon request, offering full transparency on product quality.
